One-pot synthesis of novel 2,3-dihydro-1H-indazoles.
نویسندگان
چکیده
A copper(I)-mediated one-pot synthesis of 2,3-dihydro-1H-indazole heterocycles has been developed. This synthetic route provides the desired indazoles in moderate to good yields (55%-72%) which are substantially better than those achievable with an alternative two-step reaction sequence. The reaction is tolerant of functionality on the aromatic ring.
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ورودعنوان ژورنال:
- Molecules
دوره 16 11 شماره
صفحات -
تاریخ انتشار 2011